PIPages
Labs

Vardan Karamyan

Oakland University, MI·Pharmacology

Stroke is a leading cause of death and long-term disability, and effective treatments remain scarce. One strategy is to boost the brain's own defenses after injury.

Fields

Pharmacology

Neuroscience

Biochemistry

Topics

ischemic stroke

stroke therapy

neurolysin

Grants
1 known grant, through Jun 2030

What they work on

  1. Optimize two chemical families of small-molecule activators of neurolysin (Nln), a brain-protective enzyme, to improve potency, selectivity and drug-like properties through medicinal chemistry.
  2. Determine how the activators bind and switch on neurolysin, using enzyme biochemistry and cryo-electron microscopy (cryo-EM) structures of the enzyme.
  3. Test whether optimized neurolysin activators protect the brain and support recovery in two mouse models of ischemic stroke, the type caused by blocked blood flow.

More about the research

The lab's published and pilot studies identify neurolysin (Nln) as one such defense. Nln is a peptidase, an enzyme that cuts small proteins called peptides. After stroke, Nln breaks down several peptides that harm nerve cells and produces three peptides that protect and help repair the brain. A drug that switches Nln on could therefore help the brain protect itself.

Why it matters

Many stroke patients have no effective treatment beyond restoring blood flow. Drug-like molecules that boost neurolysin, a brain enzyme that clears toxic peptides and makes protective ones, could become new medicines that limit brain damage after ischemic stroke. Learning how small molecules activate an enzyme could also guide drugs that activate other enzymes.

Known grants

From NIH and NSF research grants. Labs often have other funding we can't see.

Development and Characterization of Small Molecule Activators of Peptidase Neurolysin for Stroke Therapy

NIH · Sep 2018 – Jun 2030

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The school

Oakland University: 5 labs on PI Pages, $39M a year on research, 60 research doctorates a year.

More about Oakland University

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